Berberine and Sertraline

Supplement–drug interaction evidence from the TruthStack database.

SeverityMODERATE
Evidence TierModerate
Interaction TypeMETABOLIC
MechanismMETABOLISM
Last Reviewed2026-02-24

Summary

Berberine inhibits CYP2D6 and CYP3A4. Potential for modest increase in sertraline levels. Monitor for SSRI side effects.

CYP Enzyme Pathway Overlap

Berberine and Sertraline share activity on the following CYP enzymes:

EnzymeBerberineSertraline
CYP2D6INHIBITOR (MODERATE)SUBSTRATE (MODERATE)
CYP3A4INHIBITOR (STRONG)SUBSTRATE (WEAK)

API Reference

GET https://api.truthstack.co/v1/check?c1=Berberine&c2=Sertraline

Open, unauthenticated. Returns JSON. Developer documentation

Related Interactions

What this page is and is not. TruthStack is an informational reference database that describes published pharmacological findings. It does not provide medical advice, diagnosis, or treatment recommendations. The information on this page reflects flags in our database and should not replace consultation with a qualified healthcare provider. Always discuss supplement-drug combinations with your prescriber or pharmacist.